Global Trends in Health, Technology and Management II
Global Trends in Health, Technology and Management II
Proceedings of the 2nd International Symposium GTHTM-2025
Saxena, Anil Kumar; Saxena, Aaruni
Springer Nature Switzerland AG
02/2026
554
Mole
Inglês
9783032123190
15 a 20 dias
Descrição não disponível.
Innovations in Drug Design: Case Studies from Discovery to Development.- Development of Allosteric Inhibitors against Cyclin-Dependent Kinase 2 (CDK2).- Evaluation of 2-phenylthiazolidin-4-one analogues as inhibitors of the SARS-CoV-2 main protease.- Engineered Antibiotics: A Strategy to Combat Multi-Drug-Resistant Bacteria: A Review on Antibiotics Modification.- In silico studies of 1,2,4-triazole derivatives by targeting DHFR againsts staphylococcus aureus: Pharmacophore generation, Atom-based 3D-QSAR, Molecular docking and ADMET.- Rationale of Antifungal And Anti Bacterial Interventions Of Imidazole Derivatives.- Quantitative Structure Pharmacophore-Activity Relationship of Tricyclic Antidepressant (TCAs) Utilizing Distance-Based Features.- Computational Design of Pyrazole Derivatives for Management of Autoimmune Disease.- Designing, Synthesis and Characterization of Novel Heterocyclic Derivatives of-oxothiazolidine-3-carbonyl)-6- substituted-spiro[indoline-2,2'-thiazolidine]-3,4'-dione and -oxothiazolidine-3-carbonothioyl)-6- substituted-spiro [indoline-2,2'-thiazolidine]-3,4'-dione and their Bioevaluation.- Synthesis and Antimicrobial Evaluation of Novel dioxo spiro[indoline-3,2' thiazolidin]-3'-yl)thiourea and -dioxaspiro[indoline-3,2'-thiazolidin]-3'-yl)urea.
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Medicinal Chemistry;Drug design and development;Drug discovery;Public Health;Pharmaceutical Sciences;Artificial intelligence;Digitalization in healthcare;Sustainability;Conference Proceedings
Innovations in Drug Design: Case Studies from Discovery to Development.- Development of Allosteric Inhibitors against Cyclin-Dependent Kinase 2 (CDK2).- Evaluation of 2-phenylthiazolidin-4-one analogues as inhibitors of the SARS-CoV-2 main protease.- Engineered Antibiotics: A Strategy to Combat Multi-Drug-Resistant Bacteria: A Review on Antibiotics Modification.- In silico studies of 1,2,4-triazole derivatives by targeting DHFR againsts staphylococcus aureus: Pharmacophore generation, Atom-based 3D-QSAR, Molecular docking and ADMET.- Rationale of Antifungal And Anti Bacterial Interventions Of Imidazole Derivatives.- Quantitative Structure Pharmacophore-Activity Relationship of Tricyclic Antidepressant (TCAs) Utilizing Distance-Based Features.- Computational Design of Pyrazole Derivatives for Management of Autoimmune Disease.- Designing, Synthesis and Characterization of Novel Heterocyclic Derivatives of-oxothiazolidine-3-carbonyl)-6- substituted-spiro[indoline-2,2'-thiazolidine]-3,4'-dione and -oxothiazolidine-3-carbonothioyl)-6- substituted-spiro [indoline-2,2'-thiazolidine]-3,4'-dione and their Bioevaluation.- Synthesis and Antimicrobial Evaluation of Novel dioxo spiro[indoline-3,2' thiazolidin]-3'-yl)thiourea and -dioxaspiro[indoline-3,2'-thiazolidin]-3'-yl)urea.
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