Concepts and Models for Drug Permeability Studies

Concepts and Models for Drug Permeability Studies portes grátis

Concepts and Models for Drug Permeability Studies

Cell and Tissue based In Vitro Culture Models

Sarmento, Bruno; Leite Pereira, Catarina; Neves, Jose Das

Elsevier - Health Sciences Division

02/2024

706

Dura

Inglês

9780443155109

15 a 20 dias

Descrição não disponível.
1. Introduction
2. Importance and applications of cell- and tissue-based in vitro models for drug permeability screening in earlystages of drug development

Section I: Cell-based in vitro culture models for drug permeability studies: Immortalized and primary isolated cells
3.1. Cell-based in vitro models for buccal permeability studies
3.2. Cell-based in vitro models for gastric permeability studies
3.3. Cell-based in vitro models for intestinal permeability studies
3.4. Cell-based in vitro models for nasal permeability studies
3.5. Cell-based in vitro models for pulmonary permeability studies
3.6. Cell-based in vitro models for vaginal permeability studies
3.7. Cell-based in vitro models for transcorneal permeability studies
3.8. Cell-based in vitro models for dermal permeability studies
3.9. Tissue-based in vitro and ex vivo models for bloodebrain barrier permeability studies
3.10. Cell-based in vitro models for placental barrier permeability studies

Section II: Tissue-based in vitro and ex vivo models for drug permeability studies
4.1. Tissue-based in-vitro models for buccal permeability studies
4.2. Tissue-based in vitro and ex vivo models for intestinal permeability studies
4.3. Tissue-based in vitro and ex vivo models for nasal permeability studies
4.4. Tissue-based in vitro and ex vivo models for pulmonary permeability studies
4.5. Tissue-based models for vaginal permeability studies
4.6. Tissue-based models for ocular permeability studies
4.7. Tissue-based in vitro and ex vivo models for dermal permeability studies
4.8. Tissue-based in vitro and ex vivo models for bloodebrain barrier permeability studies Malgorzata Burek, Ellaine Salvador and Carola
4.9. Tissue-based ex vivo models for placental barrier permeability studies

Section III: Miniaturized models for drug permeability studies
5.1. Organ-on-chip models for intestinal permeability studies
5.2. Organ-on-chip models for pulmonary permeability studies
5.3. Organ-on-chip models for bloodebrain barrier permeability studies
5.4. Organ-on-chip models for other mucosal permeability studies

Section IV: Complex models for drug permeability studies
6.1. Multicompartmental dynamic models for permeability studies
6.2. Organoid-based models for permeability studies
7. Correlation between cell- and tissue-based in vitro models for drug permeability screening with in vivo situation: modeling and functional extrapolation
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Absorption; biopharmaceutics; biotechnology; bioengineering; drug development; drug transport